NK012 is a 'nanodevice' formulation of SN-38 (an irinotecan metabolite). NK012 is an SN-38-releasing polymeric micelle constructed by covalently attaching SN-38 to the block copolymer PEG-PGlu, followed by self-assembly of amphiphilic block copolymers in aqueous media.
It has completed phase II clinical trials for triple-negative breast cancer and relapsed small cell lung cancer. In 2016, Nippon Kayaku received orphan drug designation for NK012 from the US FDA. This means that if it is approved in the United States, Nippon Kayaku will be entitled to 7 years of market exclusivity. This is intended to incentivize future development, but does not mean the drug has been approved.
See also
References
- "NCI Drug Dictionary". National Cancer Institute. 2011-02-02. Retrieved 2020-11-28.
- Sumitomo; et al. (2008). "Novel SN-38–Incorporated Polymeric Micelle, NK012, Strongly Suppresses Renal Cancer Progression". Cancer Research. 68 (6): 1631–1635. doi:10.1158/0008-5472.CAN-07-6532. PMID 18339841.
- "Search of: NK012 - List Results - ClinicalTrials.gov". www.clinicaltrials.gov. Retrieved 2020-11-28.
- Nippon Kayaku Announces FDA Orphan Drug Designation to New Polymeric micelle Anti-Cancer Drug NK012 for Small Cell Lung Cancer. (2016). Evaluategroup.com. Retrieved 24 November 2017, from http://www.evaluategroup.com/Universal/View.aspx?type=Story&id=644017
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