Names | |
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IUPAC name 2-Fluoro-7H-purin-6-amine | |
Other names 2-FA | |
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3D model (JSmol) | |
ChEBI | |
ChEMBL | |
ChemSpider | |
ECHA InfoCard | 100.152.774 |
EC Number |
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PubChem CID | |
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CompTox Dashboard (EPA) | |
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Properties | |
Chemical formula | C5H4FN5 |
Molar mass | 153.120 g·mol |
Solubility in water | < 0.5 mM |
Solubility | >=10 mM in DMSO |
Hazards | |
GHS labelling: | |
Pictograms | |
Signal word | Warning |
Hazard statements | H315, H319, H335 |
Precautionary statements | P261, P264, P264+P265, P271, P280, P302+P352, P304+P340, P305+P351+P338, P319, P321, P332+P317, P337+P317, P362+P364, P403+P233, P405, P501 |
Except where otherwise noted, data are given for materials in their standard state (at 25 °C , 100 kPa). Infobox references |
2-Fluoroadenine (2-FA) is a toxic adenine antimetabolite which can be used in laboratory biological research for counterselection of wildtype bacterial or eukaryotic (i.e. animals, yeast, plants, diatoms, brown algae) APT (adenine phosphoribosyltransferase) genes. Therefore, knockouts or mutants for APT, which are resistant to 2-FA, can be selected.
2-Fluoroadenine is a critical intermediate for pharmaceutical drugs and can be synthesized within the lab from 2,6-diaminopurine, which is an inexpensive and readily available compound. In the cell, 2-Fluoroadenine is synthesized and exhibits a large range of antibacterial activity. 2-Fluoroadenine acts as an inhibitor of blood-platelet adhesion, and when combined with actinobolin, produces a greater combined effect of preventing or treating infections. In cancer treatments, 2-Fluoroadenine, has been used to treat head and neck cell carcinoma by the progressive removal of RNA and protein synthesis within tumor cells.
See also
- 5-Fluoroorotic acid (5-FOA)
References
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- "2-Fluoroadenine". pubchem.ncbi.nlm.nih.gov. Retrieved 4 May 2022.
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- Sahota, Amrik; Ranjekar, Prabhakar K.; Alfonzo, Juan; Lewin, Alfred S.; Taylor, Milton W. (1987). "Mutants of Saccharomyces cerevisiae deficient in adenine phosphoribosyltransferase". Mutation Research/Fundamental and Molecular Mechanisms of Mutagenesis. 180 (1). Elsevier BV: 81–87. doi:10.1016/0027-5107(87)90069-8. ISSN 0027-5107. PMID 3306356.
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- Serif, Manuel; Dubois, Gwendoline; Finoux, Anne-Laure; Teste, Marie-Ange; Jallet, Denis; Daboussi, Fayza (2018-09-25). "One-step generation of multiple gene knock-outs in the diatom Phaeodactylum tricornutum by DNA-free genome editing". Nature Communications. 9 (1). Springer Science and Business Media LLC: 3924. Bibcode:2018NatCo...9.3924S. doi:10.1038/s41467-018-06378-9. ISSN 2041-1723. PMC 6156588. PMID 30254261.
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- Salehi Marzijarani, Nastaran; Snead, David R.; McMullen, Jonathan P.; Lévesque, François; Weisel, Mark; Varsolona, Richard J.; Lam, Yu-hong; Liu, Zhijian; Naber, John R. (2019-08-16). "One-Step Synthesis of 2-Fluoroadenine Using Hydrogen Fluoride Pyridine in a Continuous Flow Operation". Organic Process Research & Development. 23 (8): 1522–1528. doi:10.1021/acs.oprd.9b00178. ISSN 1083-6160.
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