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Preferred IUPAC name N-(4-Aminophenyl)acetamide | |
Other names p-Aminoacetanilide, N-(4-Aminophenyl)acetamide | |
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ChemSpider | |
ECHA InfoCard | 100.004.161 |
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Properties | |
Chemical formula | C8H10N2O |
Molar mass | 150.181 g·mol |
Appearance | leaf or flake like white-Pink To Brown Powder |
Density | 1.1392 |
Melting point | 164–167 °C (327–333 °F; 437–440 K) |
Boiling point | 267 °C (513 °F; 540 K) |
Solubility in water | 0.1-1 g/100 mL at 25 °C |
Hazards | |
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Pictograms | |
Signal word | Danger |
Hazard statements | H317, H319, H334 |
Precautionary statements | P261, P264, P272, P280, P285, P302+P352, P304+P341, P305+P351+P338, P321, P333+P313, P337+P313, P342+P311, P363, P501 |
Except where otherwise noted, data are given for materials in their standard state (at 25 °C , 100 kPa). Infobox references |
4-Aminoacetanilide or paracetamin is a chemical compound which is a amino derivative of acetanilide and para-isomer of aminoacetanilide. There are two other isomers of aminoacetanilide, 2-aminoacetanilide and 3-aminoacetanilide. Aminoacetanilide derivatives are important synthetic intermediates in heterocyclic and aromatic synthesis. These derivatives have found applications in pharmaceutical industry and dyes and pigment industry.
Synthesis
Becillus cereus converts 4-phenylenediamine to 4-aminoacetanilide. Reduction of 4-nitroacetanilide by hydrogenation catalyst generates 4-aminoacetanilide. Green synthesis of p-Aminoacetanilide is achieved by reducing p-nitroaetanilide using Zn/NH4Cl in water. Number of methods are available to reduce 4-nitroacetanilide using different catalyst and reaction conditions.
Uses
4-Aminoacetanilide is used as in intermediate in the production of some dyes. 4-aminoacetanilide is also used for the synthesis of beta-lactams.
References
- ^ Singh, Raman; Kau, Rajneesh; Singh, Kuldeep (2016). "A review on Synthesis of Aminoacetanilides". Journal of Integrated Science and Technology. 4: 111–120. ISSN 2321-4635 – via Google Scholar.
- Mulyono; Takenaka, Shinji; Sasano, Yasuhiro; Murakami, Shuichiro; Aoki, Kenji (February 2007). "Bacillus cereus strain 10-L-2 produces two arylamine N-acetyltransferases that transform 4-phenylenediamine into 4-aminoacetanilide". Journal of Bioscience and Bioengineering. 103 (2): 147–154. doi:10.1263/jbb.103.147. PMID 17368397.
- 李, 玉涵; 侯, 洁; 王, 越; 吕, 连海 (2009). "催化加氢制备对氨基乙酰苯胺". 染料与染色. 46 (2): 42–45. ISSN 1672-1179.
- 曹, 玮; 曲, 波; 梁, 足培 (2004). "对氨基乙酰苯胺合成绿色工艺的研究". 化工时刊 (4): 55–56. ISSN 1002-154X.
- Gregory, Peter (2000-12-04), "Dyes and Dye Intermediates", in John Wiley & Sons, Inc. (ed.), Kirk-Othmer Encyclopedia of Chemical Technology, Hoboken, NJ, USA: John Wiley & Sons, Inc., pp. 0425051907180507.a01, doi:10.1002/0471238961.0425051907180507.a01, ISBN 978-0-471-23896-6, retrieved 2021-02-07
- Tahriri, Mozhgan; Yousefi, Mohammad; Mehrani, Kheirollah; Tabatabaee, Masoumeh; Ashkezari, Mahmood Dehghani (August 2017). "Synthesis, Characterization and Antimicrobial Activity of Two Novel Sulfonamide Schiff Base Compounds". Pharmaceutical Chemistry Journal. 51 (5): 425–428. doi:10.1007/s11094-017-1626-z. ISSN 0091-150X. S2CID 25837758.